http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2387384-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_91ce16ac3dbceb38cb5e6983c8c15a5a |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-7048 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07H17-08 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07H17-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D305-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P33-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-7048 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-04 |
| filingDate | 2000-02-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2012-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_689825bc3a4bc46032d13b8e371ba5f5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2fb99d7c27490d6ca3710629f9403b48 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_25be4daa529be870af4ae82617d431ac http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d0992b35e6e6ed8a0ec2b3ecfaa0672a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_db0db60a92587bc9a52af400ed57a37d http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f6766d4d025aeba464460b51ceadd879 |
| publicationDate | 2012-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2387384-T3 |
| titleOfInvention | Avermectin derivatives |
| abstract | A compound represented by the general formula (I) or one of its salts: wherein -X ---- Y- represents -CH> = CH-, -CH2-C (> = O) -, -CH2-CH2- or -CH2-CH (R13) -; a line ---- between R1 and a carbon atom in position 4 "represents a single or double bond; a line ---- between R2 and a carbon atom in the position represents a single or double bond; 1) when -X ---- Y- represents -CH> = CH-, the line ---- between R1 and a carbon atom at position 4 "represents a double bond; R1 represents (R11) (R12) C [wherein R11 represents a substituted or unsubstituted lower alkyl group; a formyl group; a lower alkoxycarbonyl group, the alkyl moiety of said lower alkoxycarbonyl group may be substituted with a heterocyclic group; -CH> = N-OR3, wherein R3 represents a hydrogen atom or a lower alkyl group; a lower alkenyl oxycarbonyl group; -CH> = N-NH-CONH2; a cyano group; -COR4, where R4 represents a hydroxyl group or N (R5) (R6), where R5 and R6 form a nitrogen-containing heterocyclic group together with the adjacent nitrogen atom; a vinyl group substituted with a lower alkenyl-oxycarbonyl group; - CO-S-CH2-CH2-NH-CO-Rx, wherein Rx represents a lower alkyl group; or -CH> = CH-COOH; and R12 represents a hydrogen atom or, when R11 represents a cyano group, R12 represents a hydrogen atom or a lower alkyl group]; when the line ---- between R2 and a carbon atom at position 5 represents a single bond, R2 represents a hydroxyl group, a lower alkoxy group or a tri (lower alkyl) silyloxy group; or when the line ---- between R2 and a carbon atom at position 5 represents a double bond, R2 forms a carbonyl group or a hydroxyl group (-C (> = NOH)) together with the carbon atom in the position 5.2) when -X ---- Y- represents -CH2-C (> = O) -, the line ---- between R1 and a carbon atom at position 4 "represents a double bond; R1 represents ( R11a) (R12a) C (where R11a represents a lower alkoxycarbonyl group, the alkyl moiety of said lower alkoxycarbonyl group may be substituted with a heterocyclic group or -COOCH2CH> = CH2; and R12a represents a hydrogen atom]; line ---- between R2 and a carbon atom in the position represents a single bond; and R2 represents a hydroxyl group, a lower alkoxy group or a tri (lower alkyl) silyloxy group; 3) when -X ---- Y- represents -CH2-CH2-, when the line ---- between R1 and a carbon atom at position 4 "represents a double bond, R1 represents (R11b) (R12b) C (where R11b represents to a cyano group, a carboxyl group or a lower alkenyl-oxycarbonyl group; and R12b represents a hydrogen atom]; or when the line ---- between R1 and a carbon atom at position 4 "represents a single bond, R1 can represent a carboxymethyl group or a cyanomethyl group; the line ---- between R2 and a carbon atom in position 5 represents a single bond, and R2 represents a hydroxyl group, a lower alkoxy group or a tri (lower alkyl) silyloxy group; |
| priorityDate | 1999-02-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 159.