http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2377849-T3

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04
filingDate 2008-05-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2012-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_897b45846e78f4a3f45d812330adb47d
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8268630c6f041daf5b3c4f3ddefdff58
publicationDate 2012-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2377849-T3
titleOfInvention Amino-heterocyclic compounds
abstract A compound of formula (I), or a pharmaceutically acceptable salt thereof, wherein: R is selected from the group consisting of (C1-C6) alkyl, (C2-C6) alkenyl, (C2-C6) alkynyl, cycloalkyl (C3-C8), heterocycloalkyl, aryl and heteroaryl, each of which may be optionally substituted with one to three substituents, the substituents independently selected from the group consisting of (C1-C4) alkyl, (C1-C4) alkoxy, halo and haloalkyl (C1-C4); R1 is selected from the group consisting of hydrogen, (C1-C4) alkyl, (C2-C4) alkenyl, (C2-C4) alkynyl, halo (C1-C4) alkyl and cyclopropyl; R2 is selected from the group consisting of (C1-C6) alkyl, (C2-C6) alkenyl, (C2-C6) alkynyl, (C1-C6) haloalkyl, heteroaryl selected from the group consisting of pyridinyl, pyridazinyl, pyrimidinyl and pyrazinyl , and ER5, wherein the heteroaryl may be optionally substituted with one to three substituents independently selected from the group consisting of (C1-C4) alkyl and halo (C1-C4) alkyl; R3 is selected from the group consisting of hydrogen, (C1-C4) alkyl, (C2-C4) alkenyl, (C2-C4) alkynyl, (C3-C6) cycloalkyl and (C1-C4) haloalkyl; E is selected from the group consisting of -CH2-, -CH2CH2-, -CH2CH2CH2- and -C (O) -; R5 is selected from the group consisting of cycloalkyl (C3-C8), heterocycloalkyl, aryl, aryloxy and heteroaryl, any of which may be optionally substituted with one to three substituents, such substituents being independently selected from the group consisting of (C1 -C4), alkenyl (C2-C4), alkynyl (C2-C4), hydroxyalkyl (C1-C4), haloalkyl (C1-C4), alkoxy (C1-C4), haloalkoxy (C1-C4), cycloalkyl (C3- C8), halo, cyano, phenyl, morpholinyl, (C1-C4) alkyl-amino, pyrazolyl, triazolyl and imidazolyl.
priorityDate 2007-05-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID146570
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423201936
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID197033
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID441347
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6440181
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID79033
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423201937
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423201938
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2761034
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506595
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419555681
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419546067
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID114948
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421923557
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3821
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423201640
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426117883
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54677946
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID446948
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423201641
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9896267
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419613225
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID378424
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID829861
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423201983
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19493
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70924
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4909
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450102203
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID38101
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3772069
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07943
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31244
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423201984
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420917803
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415753797
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423201997

Total number of triples: 1605.