http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2343104-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_e13cf25eb1bef6199475314477618b46 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-427 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-4184 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D235-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D277-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P19-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-427 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-437 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-422 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P37-02 |
| filingDate | 2000-04-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2010-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c2eef489deade620b5798fa9061aaf86 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d4b68ef250ceea038cf4152214b26435 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_aae3d9257e323b07864b88c07cc6fe30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b5ea93922468b75a7d8e2513f22c457b http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_71eb2f5b2f6c47082ec771f9d8fa0f38 |
| publicationDate | 2010-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2343104-T3 |
| titleOfInvention | AMINA DERIVATIVES |
| abstract | An amine-derived compound of the formula (I): ** (See formula) ** in which: R1 represents a carbamoyl group (which may have one or two α substituents described below), a thiocarbamoyl group (which may have one or two α substituents described below) or a sulfonyl group (having an α substituent described below); each R2 and R3 represents a hydrogen atom, a C1-C10 alkyl group, a C6-C10 aryl group (which may have 1 to 3 β substituents described below) or a C7-C16 aralkyl group (which may have 1 to 3 β substituents described below in the aryl portion); each W1, W2 and W3 represents a single bond or a C1-C8 alkylene group; each X, Y and Q represents an oxygen atom or a sulfur atom; Z represents a group = CH- or a nitrogen atom; Ar represents a benzene ring or a naphthalene ring; L represents 1 to 4 substituents on the Ar ring and the or each substituent is a hydrogen atom, a C1-C6 alkyl group, a C6-C10 aryl group (which may have 1 to 3 β substituents described below) or a C7-C16 aralkyl group (which may have 1 to 3 β substituents described later in the aryl portion); the substituent α represents (i) a C1-C10 alkyl group, (ii) a C1-C6 haloalkyl group, (iii) a C3-C10 cycloalkyl group, (iv) a C6-C10 aryl group (which may have 1 to 3 γ substituents described below), (v) a C7-C16 aralkyl group (which may have 1 to 3 γ substituents described below in the aryl portion), (vi) a C4-C11-carbonyl cycloalkyl group, (vii ) a C7-C11 arylcarbonyl group (which may have 1 to 3 γ substituents described later in the aryl portion), (viii) a C8-C17 aralkylcarbonyl group (which may have 1 to 3 γ substituents described later in aryl portion), (ix) an aromatic heterocyclic group (which may have 1 to 3 γ substituents described below), (x) an aromatic heterocyclic carbonyl group (which may have 1 to 3 γ substituents described below), ( xi) a C1-C6 alkylsulfonyl group, (xii) a C1-C6 halogenoalkylsulfonyl group, (xiii) a C6-C10 arylsulfonyl group (which it may have 1 to 3 γ substituents described below in the aryl portion), or (xiv) a C7-C16 aralkylsulfonyl group (which may have 1 to 3 γ substituents described later in the aryl portion); the substituent β represents (i) a C1-C6 alkyl group, (ii) a C1-C6 halogenoalkyl group, (iii) a C1-C6 alkoxy group, (iv) a halogen atom, (v) a hydroxyl group, ( vi) a C6-C10 aryl group (which may have 1 to 3 δ substituents described below), (vii) a C7-C16 aralkyl group (which may have 1 to 3 δ substituents described later in the aryl portion) , (viii) a cyano group, (ix) a nitro group, or (x) an amino group (which may have one or two δ substituents described below); the γ substituent represents (i) a C1-C6 alkyl group, (ii) a C1-C6 haloalkyl group, (iii) a C1-C6 alkoxy group, (iv) a halogen atom, (v) a hydroxyl group, ( vi) a cyano group, (vii) a nitro group, (viii) a C3-C10 cycloalkyl group, (ix) a C6-C10 aryl group (which may have 1 to 3 C1-C6 alkyl groups, C1- haloalkyl groups C6, C1-C6 alkoxy groups or halogen atoms as substituents), (x) a C7-C16 aralkyl group (which may have 1 to 3 C1-C6 alkyl groups, C1-C6 haloalkyl groups, C1-C6 alkoxy groups or halogen atoms as substituents on the aryl moiety), (xi) a C1-C7 aliphatic acyl group, (xii) a C1-C7 aliphatic acyloxy group, (xiii) an amino group, (xiv) a di- (C1-alkyl group) -C6) amino or (xv) a C1-C4 alkylenedioxy group; the substituent δ represents (i) a C1-C10 alkyl group, (ii) a C6-C10 aryl group (which may have 1 to 3 C1-C6 alkyl groups, C1-C6 halogenoalkyl groups, C1-C6 alkoxy groups or atoms halogen as substituents), (iii) a C7-C16 aralkyl group (which may have 1 to 3 C1-C6 alkyl groups, C1-C6 haloalkyl groups, C1-C6 alkoxy groups or halogen atoms as substituents on the aryl portion ), (iv) a C1-C7 aliphatic acyl group, (v) a C4-C11 cycloalkylcarbonyl group, (vi) a C7-C11 arylcarbonyl group (which may have 1 to 3 C1-C6 alkyl groups, C1- haloalkyl groups C6, C1-C6 alkoxy groups or halogen atoms as substituents), (vii) a C8-C17 aralkylcarbonyl group (which may have 1 to 3 C1-C6 alkyl groups, C1-C6 halogenoalkyl groups, C1-C6 alkoxy groups or halogen atoms as substituents on the aryl moiety), (viii) an aromatic heterocyclic carbonyl group (which may have 1 to 3 C1-C6 alkyl groups, halogenoal groups C1-C6 alkyl, C1-C6 alkoxy groups or halogen atoms as substituents); or a pharmaceutically acceptable salt thereof. |
| priorityDate | 1999-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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