http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2327210-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_b9237fdf6dca9ac365fc5166858e7862 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-14 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B61-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-505 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-506 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-14 |
| filingDate | 2001-07-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2009-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e201c7dc269302774d33989fc7b0fd69 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a9125530d0ad8a2d919e2484d8ce5117 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b83456c48abe2f5a3cdbebf1a90de59c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_09e39e4cefb2ff9c98a5083f1088dd99 |
| publicationDate | 2009-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2327210-T3 |
| titleOfInvention | DERIVATIVES OF VARIOLINA AS ANTI-BANERIGAN AGENTS. |
| abstract | Compound of formula (I): ** see formula ** in which: R1 and R2 are each independently selected from the group consisting of H, OH, OR '', SH, SR '', SOR '', SO2R ' ', NO2, NH2, NHR' ', N (R' ') 2, NHCOR' ', N (COR' ') 2, NHSO2R' ', CN, halogen, C (= O) H, C (= O) R '', CO2H, CO2R '', C1-C12 alkyl, C1-C12 haloalkyl, C2-C12 alkenyl, C2-C12 alkynyl, substituted or unsubstituted aryl, substituted or unsubstituted aralkyl and substituted or unsubstituted heteroaromatic group; and R3 is selected from the group consisting of OH and OMe; wherein the or each group R '' is independently selected from the group consisting of OH, C1-C12 alkyl, C1-C12 haloalkyl, C2-C12 alkenyl, C2-C12 alkynyl, substituted or unsubstituted aryl, substituted or unsubstituted aralkyl substituted, substituted or unsubstituted arylalkenyl and substituted or unsubstituted heteroaromatic group, and wherein when the group R1 or R2 is a group of formula N (R '') 2 or N (COR '') 2, each of the R groups "may be the same or different, or the two R groups", together with the nitrogen atom to which they are attached, may form a 5-14 membered heterocyclic ring; the aryl group and the aryl moiety of the aralkyl and arylalkenyl group are a carbocyclic aryl group having from 6 to 14 carbon atoms in a carbocyclic ring or two or more condensed rings; the aralkyl group is a C1-C6 alkyl group that is substituted with an aryl group as defined above; the arylalkenyl group is a C2-C6 alkenyl group that is substituted with an aryl group as defined above; the heteroaromatic group is a heterocyclic aromatic group having from 5 to 14 ring atoms in a ring or two or more condensed rings from which at least one ring atom is selected from the group consisting of nitrogen, oxygen and sulfur, and a heterocyclic aromatic group of this type fused to an aryl group as defined above; the substituents on the aryl and heteroaromatic groups and the aryl moiety of the aralkyl and arylalkenyl groups are selected from the group consisting of C1-C12 alkyl, C1-C12 haloalkyl, C1-C12 alkoxy, C1-C12 alkylthio, NH2, C1- alkylamino C4, di (C1-C4 alkyl) amino, C1-C4 alkanoylamino, di (C1-C4 alkanoyl) amino, NO2, CN and halogen; and wherein one or more of the tertiary amine nitrogen atoms of formula (I) are optionally quaternized, and salts and esters thereof, with the exception of the compounds in which: R1 and R2 are amino and R3 is hydroxyl . |
| priorityDate | 2000-07-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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