http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2322727-A1

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filingDate 2005-07-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_111b2144b9f7f41ad55908fd79cf9492
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0e555d87a14bd3ea90be63dace447669
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publicationDate 2009-06-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2322727-A1
titleOfInvention METHOD FOR QUANTIFYING THE PROTEIN G COUPLED RECEPTOR UNION (GPCR) -PROTEIN G BY USING A CELL MEMBRANE ARRAY.
abstract Method to quantify receptor bindingncoupled to protein G (GPCR) -protein G by thenuse of an array of cell membranes.n n n The method comprises (i) contacting anunmarked candidate compound with an array of cell membranesnin the presence of labeled GTP or an analogue thereof, nonhydrolysable, marked, under conditions that allow interactionnbetween said compound and said GPCR present in said membranesncellular, and between said labeled or analog GTP thereof and saidnG protein present in said membranes; (ii) wash; and (iii)nquantify the signal obtained by the union of the GTP (or analog)nlabeled to said protein G. Of application in the analysis of theninteraction between compounds and membrane receptor proteinsncellular and intracellular signaling mechanisms thatntriggers this mechanism of interaction mediated by saidncompounds.
priorityDate 2005-07-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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