http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2318284-T3

Outgoing Links

Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_1b0c198757da18cf77dfbdcef00abb70
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-64
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-08
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-24
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-48
filingDate 2004-04-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2009-05-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3b5634f8ac262d040e41e7d2120eee45
publicationDate 2009-05-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2318284-T3
titleOfInvention ANALOG OF THE GONADOTROPIN HORMONE CONJECTED WITH STEROID HORMANS.
abstract A compound consisting of a gonadotropin-releasing hormone analogue (GnRH) conjugated to a portion of steroid hormone, or a C11, C17 or C21 hydroxy derivative thereof, which is capable of binding to a hormone binding protein plasma selected from cortisol binding globulin (CBG), sex hormone binding globulin (SHBG) and albumin, in which the GnRH analog is a GnRH antagonist selected from [AcD-Nal 1, D-Cpa 2, D-Pal 3, Arg 5, D-Lys 6, D-Ala 10] GnRH, [Ac-deltaPro 1, D-Fpa 2, D-Trp 3, D-Lys 6] GnRH, Cetrorelix, Ganirelix, Abarelix , Antide, Teverelix, FE200486, Na-Glu, A-75998, A-76154, A-84861, D-26344, D-63153, D21775, ramorelix, degarelix, NBI-42902, Org-30850, detirelix, iturelix, TAK -013, TAK810, AN 207, AcD-Nal-D-Cpa-D-Pal-Ser-Arg-D-Lys-Leu-Arg-Pro-D-Ala-NH2; Ac-deltaPro-D-Fpa-D-Trp-Ser-Tyr-D-Lys-Leu-Arg-Pro-Gly-NH2; AcD-Nal-D-Cpa-D-Pal-Ser-Arg-D-Lys-Lys-Leu-Arg-D-Ala-NH2; D-Pal-Ser-Arg-D-Lys-Leu-Arg-Pro-D-Ala-NH 2; AcD-Nal-D-Cpa-D-Pal-Ser-Arg-D-Lys-Lys-Arg-Pro-D-Ala-NH 2; [D-Pyr 1, D-Phe 2, D-Trp 3-6] GnRH; D-Lys 6 Antide; Lys 5 Antide or Lys 8 Antide, or a GnRH agonist selected from pGlu-His-Trp-Ser-Tyr-D-Lys-Leu-Arg-Pro-GlyNH2, Triptorelin, Buserelin, leuprolide, goserelin, deslorelin, ProMaxx- 100, avorelin, histrelin, nafarelin, leuprorelin or triptorelin.
priorityDate 2003-04-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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