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filingDate 2001-03-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2009-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_470954e4e91413e19a6a94dc384a4447
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publicationDate 2009-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2311012-T3
titleOfInvention DOPAMINE D3 RECEIVER LINKS FOR THE ADDICTION TREATMENT.
abstract Use of the compounds, which are chosen from 2 - [(3- {4- [2-tert-butyl-6- (trifluoromethyl) -4-pyrimidinyl] -1-piperazinyl} propyl) -sulfanyl] -4- pyrimidinol, 5 - ({3- [4- (3,5-dichlorophenyl) -1-piperazinyl] propyl} sulfanyl) -1,3,4-thiadiazol-2-amine, 5 - [(2-methyl- 3- (4- [3- (trifluoromethyl) phenyl] -1-piperazinyl) propyl) sulfanyl] -1,3,4-thiadiazol-2-amine, 2 - [{3- (4- [3- (trifluoromethyl) ) phenyl] -1-piperazinyl} propyl) sulfanyl] -4-pyrimidinol, 5- (6- {4- [3- (trifluoromethyl) phenyl] -1-piperazinyl) hexyl) -1,3,4-thiadiazole- 2-amine, 1 - {(2E) -4 - [(4-hydroxy-2-pyrimidinyl) sulfanyl] -2-butenyl} -4- [3- (trifluoromethyl) phenyl] piperazindiium, 4-methyl dichloride -5 - [(3- (4- [3- (trifluoromethyl) phenyl] -1-piperazinyl) propyl) sulfanyl] -4H-1,2,4-triazol-3-amine, 2 - ([3- ( 4- [3- (trifluoromethyl) phenyl] -3,6-dihydro-1 (2H) -pyridinyl) propyl] sulfanyl) -4-pyrimidinol, 2 - ({3- [4- (3-isopropylphenyl) -1 -piperazinyl] propyl} sulfanyl) -4-pyrimidinol, 5 - [(3- {4- [6- (trifluoromethyl) -2-pyridinyl] -1-piperazinyl} propyl) sulfanyl} -1,3,4-thiadiazole -2-ami na, 5 - [((2E) -4- (4- [6- (trifluoromethyl) 2-pyridinyl] -1-piperazinyl) -2-butenyl) sulfanyl] -1,3,4-thiadiazol-2-amine , 5 - ({3- [4- (3,5-diterc.-butylphenyl) 1-piperazinyl] propyl} sulfanyl) -4-methyl-4H-1,2,4-triazol-3-amine, - ({7- [4- (3-Isopropylphenyl) -1-piperazinyl] heptyl} sulfanyl) -1,3,4-thiadiazol-2-amine, 4-ethyl-5 - [(3- (4- [ 3- (trifluoromethyl) phenyl] -1-piperazinyl) propyl) sulfanyl] -4H-1,2,4-triazol-3-amine, 3- (4- {8 - [(5-amino-1,3, 4-thiadiazol-2-yl) sulfanyl] octyl) -1-piperazinyl) -benzonitrile, 5 - [(3- (4- [6-methyl-2- (1H-pyrrol-1-yl) -4-pyrimidinyl) ] -1-piperazinyl} propyl) -sulfanyl] -1,3,4-thiadiazol-2-amine, 4-methyl-5 - [(3- {4- [6-methyl-2- (1H-pyrrole- 1-yl) -4-pyrimidinyl] -1-piperazinyl} -propyl) sulfanyl] -4H-1,2,4-triazol-3- amine, the 5 - [{(2E) -4- (4- [2 -terc.-butyl-6- (trifluoromethyl) -4-pyrimidinyl] -1-piperazinyl) -2-methyl-2-butenyl} sulfanyl] -4-methyl-4H-1,2,4-triazol-3-amine , 1- [3- (difluoromethyl) phenyl) -4- (3 - ([4-methyl-5- (methylammonium) -4H-1,2,4-triazol-3-yl] sulfanyl) propyl) dichloride piperazin- 4-io and the 5 - ({3- [4- (2,6-diterc.-butyl-4-pyrimidinyl) -1-piperazinyl] propyl} sulfanyl) -1,3,4-thiadiazol-2-amine, or its salts with physiologically compatible acids, to obtain a drug for the treatment of addiction.
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