abstract |
A TRICYCLE COMPOUND OF THE GENERAL FORMULA (I) AS DEFINED HEREIN WHICH PRESENTS AN ANTAGONIST ACTIVITY TO RECEPTORS V {SUB, 1} AND / OV {SUB, 2} AND PRESENTS AN INTAGONIST ACTIVITY IN VIVO TO VASOPRESIN, METHODS FOR USE OF SUCH COMPOUNDS IN THE TREATMENT OF DISEASES CHARACTERIZED BY A RENAL REABSORTION IN EXCESS OF WATER AND A PROCESS FOR THE PREPARATION OF SUCH COMPOUNDS. |