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filingDate 2003-04-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3fd9d5c622f1b407dd9c6981134df51d
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publicationDate 2005-06-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2234393-A1
titleOfInvention "FORMULATIONS OF PELETS OF BENCIMIDAZOLIC COMPOUNDS ANTIULCEROSOS AND LABILES TO THE ACID".
abstract Compound pellet formulationsnbenzimidazole antiulcer and acid labile.n n n They comprise inert sugar / starch granules thatnare: initially coated with an active and non-alkaline layernwhich has the benzimidazole compound (omeprazole, lansoprazole,npantoprazole, rabeprazole, etc.), sodium and / or potassium salts ofnacids of formula R-O-SO 3 Hnwhere R is a fatty acid alkyl radicaln(C 6 -C 20) (preferably lauryl sulfatensodium), fatty acids (C 6 -C 20)n(preferably oleic acid), sodium and / or potassium salts ofn(C 6 -C 20) fatty acids (preferablynpotassium oleate), sodium carboxymethylcellulose andnpolyvinylpyrrolidone; second coated with a non-layernseparation alkaline having hydroxypropyl methylcellulose; Ynfinally coated with an enteric layer. Molar relationshipnPreferred (sodium lauryl sulfate): (oleic acid + potassium oleate)nIt is between 4: 1 and 6: 1. All coatings are made withnaqueous solutions, suspensions or dispersions at a temperaturenrelatively high, and all drying is done at temperaturenrelatively low and for a relatively short time. They arenstable over time and useful for oral administration.
priorityDate 2003-04-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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