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publicationDate 2005-03-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2225103-T3
titleOfInvention NEW LHRH ANTAGONISTS WITH IMPROVED DISSOLUTION PROPERTIES.
abstract Compounds of the general formula 1 A-Xxx1-Xxx2-Xxx3-Xxx4-Xxx5-Xxx6-Xxx7-Xxx8-Xxx9-Xxx10- NH2 in which they mean an acetyl group or a 3- (4-fluorophenyl) group - propionyl Xxx1 D-Nal (1) or D-Nal (2), Xxx2-Xxx3D-Cpa-D-Pal (3) or a single link, Xxx4 Ser, Xxx5 N-Me-Tyr, Xxx6 D-Hci, Xxx7 Nle, Xxx8 Arg or Lys (iPr), Xxx9 Pro, and Xxx10 Ala or Sar and their salts with pharmaceutically acceptable acids.
priorityDate 1999-03-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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