http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2213044-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_34bd4e87ecbca17f16d460ca394e60f9 |
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C40B40-00 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C40B40-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-6561 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 |
| classificationIPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B61-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-435 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-437 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D513-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K48-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/B29D30-52 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F9-6561 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4745 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-53 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-519 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/G11C29-00 |
| filingDate | 2000-09-18-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2004-08-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_82f1a68006ba3a54ac1d5c6000613cf5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_95be756c16a65fd7da0cc795ea35f364 |
| publicationDate | 2004-08-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2213044-T3 |
| titleOfInvention | NEW IMIDAZO-3-IL-BICYCLE AMINES. |
| abstract | Bicyclic imidazo-3-yl-amines of general formula I, in which X represents CR4 or N and Y represents CR5 or N, with the proviso that X and Y do not mean simultaneously N, R1 represents (CH2) nCN with n = 4, 5 or 6, if necessary substituted phenyl, C4-C8-cycloalkyl, CH2CH2R (R = 4-morpholino), 1, 1, 3, 3-tetramethyl-butyl or CH2Ra, where Ra is equal to hydrogen, OH, C1 -C8-alkyl (branched or unbranched), substituted phenyl, CO (OR '') (with R '' = C1-C4-unbranched alkyl or C1-C5-branched alkyl), PO (OR '' ) 2 (with R '' = C1-C4-unbranched alkyl or C1-C5-branched alkyl) or Si (RxRyRz) (Rx, Ry and Rz being in each case, independently of each other, C1-C4-alkyl (branched or unbranched), C4-C8-cycloalkyl or phenyl), R2 represents hydrogen, CORb, Rb being equal to C1-C4-alkyl (branched or unbranched) or C3-C8-cycloalkyl, CH2CH2CO (ORc), Rc being the same to C1-C4-alkyl (branched or unbranched), adamantyl, phenyl, if substituted, 1- naphthyl or 2-Naphthyl, if substituted, or 2-pyridyl, 3-pyridyl, 4-pyridyl, thiazolyl or furoyl, optionally substituted in each case, CH2-phenyl, CH2CH2Rd, where Rd is equal to phenyl if substituted, or CONHRe, being Re equal to C1-C80-alkyl (branched or unbranched), C3-C8-cycloalkyl or phenyl if substituted, R3 represents C1-C8-alkyl (branched or unbranched), C3-C8-cycloalkyl, phenyl in case substituted die, naphthyl if substituted, pyrrole if substituted, pyridyl if substituted, furan if substituted, thiophene if substituted, anthracene if substituted, phenanthrene, if substituted, or quinoline if substituted , R4, R5, R6 and R7 are selected from the group consisting of hydrogen, NO2, NH2, OH, CF3, Cl, F, Br, CN, methyl or OR '' '', where R '' '' = benzyl, or R6 and R7 together form a bridge -CH = CH-CH = CH- and residues R4 and R5, if they exist, represent hydrogen, with the proviso that as at least one of the residues R4, R5, R6 or R7 present in the molecule is not hydrogen and, when R1 means methyl, ethyl, propyl, n-butyl, isobutyl, CO (O-methyl) or benzyl, R3 is not methyl, and , when one of the residues R4, R5, R6 and R7 means O-benzyl or R4 means OC1-C4-alkyl (branched or unbranched), R1 is not CH2Ra (being Ra hydrogen or C1-C5-alkyl (branched or not branched)), in the form of pharmaceutically acceptable bases or salts. |
| priorityDate | 1999-10-08-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
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