abstract |
A SERIES OF CIS -3 [ARYLMETHYL (SUBSTITUTED ALPHA)] QUINUCLIDINES, 3- [METHYLAMINE (CYCLIC)] AND ACUTEALLY ACCEPTABLE CIS IS PRESENTED. THESE PARTICULAR COMPOUNDS ARE USEFUL AS ANTAGONISTS P AND ALSO, HAVE GREAT VALUE IN THE TREATMENT OF GASTROINTESTINAL DISEASES, DISEASES OF THE CENTRAL NERVOUS SYSTEM, INFLAMMATORY DISEASES OR PAIN OR MIGRAINE. PREFERRED COMPOUNDS INCLUDE ETHYLAMINE CIS ((2-TRIFUOROPHENYL)] CIS METHODS ARE ALSO SUPPLIED TO PREPARE THESE COMPOUNDS FROM KNOWN INITIATOR MATERIALS. |