http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3896062-A1

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filingDate 2019-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_adcd42ee994a8e8fa597130afdeae8cd
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publicationDate 2021-10-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3896062-A1
titleOfInvention Isoindoline compound, and preparation method, pharmaceutical composition, and application of isoindoline compound
abstract The present invention relates to an isoindoline compound as represented by general formula (I) and used as a CRBN regulator, and a preparation method, a pharmaceutical composition, and an application of the isoindoline compound. Specifically, a class of polysubstituted isoindoline compound provided in the present invention, as a class of CRL4<sup>CRBN</sup> E3 ubiquitin ligase regulator having a novel structure, has good anti-tumor activity and immunoregulatory activity, and can be used for preparing drugs for treating diseases associated with a CRL4<sup>CRBN</sup> E3 ubiquitin ligase.
priorityDate 2018-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 2158.