http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3863720-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-4545
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filingDate 2019-10-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f7438ae294583211289424ce1d7fc7c6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_797e47cbb100210dec3c671a93cdcba0
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publicationDate 2021-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3863720-A1
titleOfInvention Small molecule mdm2 protein degraders
abstract The present disclosure provides compounds represented by Formula (I): wherein R la , R lb , R 2a , R 2b , R 3a , R 3b , R 4 , A, L, X, Y, and Z are as defined as set forth in the specification. The present disclosure also provides compounds of Formula (I) for use to treat cancer or any other disease, condition, or disorder that is responsive to degradation of MDM2 protein.
priorityDate 2018-10-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395394
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID460612
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0CN75
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21329
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226414652
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226458111
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5073
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22513
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865C5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9V1P1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ01558
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396787
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5070
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395401
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0CE13
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID36314
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID644241
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID56487
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1RV79
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87057646
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15324
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6442177
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2083
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31703
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395361
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2907
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395360
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393605
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21328
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID656583
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID446512
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00356
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8PTD3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID80604
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00355
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226421412
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397750
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID30590
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID540378
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID472335
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397688
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395327
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7157
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID13645
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395705
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119031
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0R2M2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00362
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395359
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID9048
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ90YK5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00361
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24664
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4336216
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5035
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396694
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID938
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395352
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100052545
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3152
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP32809
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6VIW4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6A548
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2662
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397640
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400055
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395706
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID536642
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281845
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID443939
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID32191
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1KVQ9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5359013
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID35728
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395633
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID131986901
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5JHB5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66616196
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395318
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97399
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395833
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16858
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID852825
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395832
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCAAB71619
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151194
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23916
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151193
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408924
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396627
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395836
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396623
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID41230
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395835
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID408035
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24481
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281542
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4WVG0
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395834
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA2BLC6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6400441
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6URW1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226416012
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126941
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23722
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100009074
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226471570
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24383
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5978
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151166
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO34425
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393257
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6UUN9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399873
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8892
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP62975
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID111332
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119607
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393245
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP75358
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399864
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO32755
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5979
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399201
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID58799
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9YFS9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60953
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226420957
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4340567
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135398745
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCE2RST8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395748
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17246
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226420956
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13678
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2187
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25313
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ71RP1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID38769
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID196
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83348
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP97793
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID36462
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135398658
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226530364
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119570
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HSS7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ94469
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399863
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO28542
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60937
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25589
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395766
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO14746
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136187588
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ94819
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID249332
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399177
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID216818
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226432694
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14985
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83456
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ94818
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395715
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15550481
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11682
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP17721
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397441
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID45051774
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31307
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HJ69
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59693

Total number of triples: 812.