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filingDate 2019-08-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8a269763c59bbe961048865a69c2a5d0
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publicationDate 2021-07-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3844190-A1
titleOfInvention Methods and compounds for targeting sortilin receptors and inhibiting vasculogenic mimicry
abstract The present disclosure relates to peptide compounds and conjugate compounds, processes, methods and uses thereof for treatment of cancer or aggressive cancer. For example, the compounds can comprise compounds of formula X1 X2X3X4X5GVX6AKAGVX7NX8FKSESY (I) (SEQ ID NO: 1) (X9)nGVX10AKAGVX11NX12FKSESY (II) (SEQ ID NO: 2) YKX13LRRX14APRWDX15PLRDPALRX16X17L (III) (SEQ ID NO: 3) YKX18LRR(X19)nPLRDPALRX20X21L (IV) (SEQ ID NO: 4) IKLSGGVQAKAGVINMDKSESM (V) (SEQ ID NO: 5) IKLSGGVQAKAGVINMFKSESY (VI) (SEQ ID NO: 6) IKLSGGVQAKAGVINMFKSESYK (VII) (SEQ ID NO: 7) GVQAKAGVINMFKSESY (VIII) (SEQ ID NO: 8) GVRAKAGVRNMFKSESY (IX) (SEQ ID NO: 9) GVRAKAGVRN(Nle)FKSESY (X) (SEQ ID NO: 10) YKSLRRKAPRWDAPLRDPALRQLL (XI) (SEQ ID NO: 11) YKSLRRKAPRWDAYLRDPALRQLL (XII) (SEQ ID NO: 12) YKSLRRKAPRWDAYLRDPALRPLL (XIII) (SEQ ID NO: 13) wherein X1 to X21 and n can have various different values and wherein at least one protecting group and/or at least one labelling agent is optionally connected to said peptide compound at an N- and/or C-terminal end, for use in inhibiting vasculogenic mimicry and/or for treating a cancer.
priorityDate 2018-08-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6V919
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409204
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A038
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WN83
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18477222
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO28542
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226449222
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14242
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID445154
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5429
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60700
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22513
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226513570
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ64191
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114401
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397873
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395931
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID457193
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP32809
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF6RKC1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1794427

Total number of triples: 638.