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filingDate 2019-07-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_25d9c6a529ee7f80d7b0160163d301d3
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publicationDate 2021-05-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3820473-A1
titleOfInvention Enzymatic synthesis of 4'-ethynyl nucleoside analogs
abstract The present invention relates to an enzymatic synthesis of 4'-ethynyl-2'-deoxy nucleosides and analogs thereof, for example EFdA, that eliminates the use of protecting groups on the intermediates, improves the stereoselectivity of glycosylation and reduces the number of process steps needed to make said compounds. It also relates to the novel intermediates employed in the process.
priorityDate 2018-07-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393686
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3P7M3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7N932
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ668Z0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9CB45
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP44406
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8K9W6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9PPQ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3L0F7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9PPP3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0UTU0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO32808
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP57526
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5988
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID104815
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226496689
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO24821
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68906
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68905
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6NF47
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9C2U0

Total number of triples: 1916.