http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3705471-A1

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filingDate 2018-11-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8d0f7698e89adaf560c2d1f7adc71222
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publicationDate 2020-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3705471-A1
titleOfInvention Double-headed protease inhibitor
abstract The present invention provides a compound that is highly safe and useful in the prevention, alleviation, and/or treatment of various diseases involving enteropeptidase inhibition and/or trypsin inhibition, a pharmaceutical composition containing the compound, a method for producing the compound, and the like. Specifically, the present invention provides a compound represented by the following general formula (I):[wherein: A<sup>1</sup>and A<sup>2</sup>each independently represent an inhibitor residue having at least one activity selected from an enteropeptidase inhibitory activity and a trypsin inhibitory activity; and Z represents a spacer that links A<sup>1</sup>to A<sup>2</sup>] or a pharmaceutically acceptable salt thereof.
priorityDate 2017-11-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465249338
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155093565
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465281662
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311736856
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311736841
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID518121
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155093674
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10632253
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155093651
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155093516
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311406682
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123262618
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311406683
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Total number of triples: 1758.