http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3652184-A1

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publicationDate 2020-05-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3652184-A1
titleOfInvention Macrocyclic mcl-1 inhibitors and methods of use
abstract The present invention relates to compounds of the formula (I), wherein A 2 , A 3 , A 4 , A 6 , A 7 , A 8 , A 15 , R A , R 5 , R 9 , R 10A , R 10B , R 11 , R 12 , R 13 , R 14 , R 16 , W, X, and Y have any of the values defined in the description, as well as pharmaceutical grade salts thereof, which are usable as agents in the treatment of diseases and conditions, including cancer. The present invention further relates to pharmaceutical compositions comprising the compounds of formula (I).
priorityDate 2017-08-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 821.