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filingDate 2018-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2020-04-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3643704-A1
titleOfInvention New intermediates for the preparation of remifentanil hydrochloride
abstract A new intermediate for synthesizing 1-substituted-4-[phenyl(propanoyl)amino]piperidine-4-carbonitrile derivatives is laid open. Specifically set out is a method for use of this intermediate in the preparation of remifentanil. The enclosed shorter process offers a greater yield of products with higher purity as compared to methods reported in the prior art.
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