http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3532056-A1

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filingDate 2017-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1a5887ff021d0de1a314332cea28f4bb
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7fadc00e809383c457c8b294f7d8c7d4
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publicationDate 2019-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3532056-A1
titleOfInvention Aldosterone synthase inhibitor
abstract The present invention relates to a compound selected from (R)-(+)-5-(p-cyanophenyl)- 5,6,7,8-tetrahydroimidazo[1,5-a]pyridine and a pharmaceutically acceptable salt thereof, and in particular to the phosphate salt of (R)-(+)-5-(p-cyanophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine, both having preferably an enantiomeric excess of the (R) form higher than or equal to 97%. Furthermore, the present invention relates to pharmaceutical compositions comprising the same, their use as a medicament and in methods of treatment of diseases and disorders in humans including women of child bearing potential and pediatric patients in which aldosterone over-exposure contributes to the deleterious effects of said diseases or disorders, as well as processes for preparing said inventive compounds.
priorityDate 2016-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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