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filingDate 2017-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_dde74f781c2f68e8b7e015e981b1e936
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publicationDate 2019-04-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3464286-A1
titleOfInvention Pyrazolopyridine derivatives for the treatment of cancer
abstract The present invention relates to a compound formula (I): and to salts thereof, wherein R 1 , R 2 X, and Y have any of the values defined herein, and compositions and uses thereof. The compounds are useful as inhibitors of CBP and/or EP300. Also included are pharmaceutical compositions comprising a compound of formula (I) or a pharmaceutically acceptable salt thereof, and methods of using such compounds and salts in the treatment of various CBP and/or EP300-mediated disorders such as cancer, inflammatory disorders and autoimmune diseases.
priorityDate 2016-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396574
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394558
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169494
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169505
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396545
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57504783
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227399590
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID50294
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID50295
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396540
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396158
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316757431
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID441409
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396155
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID27447
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284365
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408415
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132168841
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396151
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394498
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408367
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226417921
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60871
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169483
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4033
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169484
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24847774
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394363
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394364
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409017
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169463
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169464
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2792
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID104741
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2725
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169462
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID273286
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226418074
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169459
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4044
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17986852
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396117
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169460
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132168842
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423521
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733525
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394420
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132168843
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226413443
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733526
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169474
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423478
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4037
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID43806
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132168821
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60877
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2832
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6436
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396111
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID688461
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID42609283
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132168820
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16702
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394385
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393293
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57006608
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4432299
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57453785
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226413489
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132168830
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID443958
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396123
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID443943
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169446
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132168828
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2791
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60852
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2265
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15700889
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24871113
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169457
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226453864
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132169456
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2776
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5503
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Total number of triples: 2050.