http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3404026-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-519
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-519
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-04
filingDate 2016-12-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_24b5c1218341119778f66723c9a230ac
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3e6be8c645d9907d6f2dea45b9bff3e8
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_87aa833fcaf20ef426f237b22c5dd5fa
publicationDate 2018-11-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3404026-A1
titleOfInvention Pyrimido-isoquinolin-quinone derivative compounds, and pharmaceutically acceptable salts, isomers and tautomers thereof; pharmaceutical composition; preparation method; and use thereof in the treatment of diseases caused by bacteria and multidrug-resistant bacteria
abstract The present invention provides pyrimidine-isoquinolin-quinone derivatives of formula I, their salts, isomers, pharmaceutically acceptable tautomers; pharmaceutical composition; preparation procedure; and their use in the treatment of bacterial and resistant bacterial diseases, such as methicillin-resistant Staphylococcus aureus (MRSA), intermediate vancomycin-resistant Staphylococcus aureus (VISA), vancomycin-resistant Staphylococcus aureus (VRSA), vancomycin-resistant Enterococcus spp. (VRE), Enterococcus faecalis, Emerging Staphylococcus aureus with resistance to linezolid and/or bacterial strains not susceptible to daptomycin.n nWhere the radicals R 1 , R 2 , R 3 , R 4 and R 5 are as defined in the work specifications of the present invention.
priorityDate 2015-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377368
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226433937
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID240147
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377357
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226495186
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344146300
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377359
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12765
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344146304
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66049
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID130204570
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344146305
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID243
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344146642
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394361
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226411107
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17882607
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID81152
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377582
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19066652
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377584
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11276017
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344147005
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377576
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344147006
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377577
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226674112
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377337
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID377293819
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344147007
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377578
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377338
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226514812
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID377293822
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344147008
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377579
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377339
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID377293823
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344146644
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377592
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377340
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID84989
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID377293824
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344147001
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396344
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID377293650
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344147002
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135377599

Total number of triples: 351.