http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3322701-A1

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filingDate 2016-07-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_db25eaec2b018021208e3d834d76fa52
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publicationDate 2018-05-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3322701-A1
titleOfInvention Ethynyl derivatives as metabotropic glutamate receptor modulators
abstract The present invention relates to compounds of formula I wherein R 1 is lower alkyl; R 2 is phenyl or pyridinyl, wherein the N atom in the pyridinyl group may be in different positions; n is 0, 1 or 2; V/U are independently from each other O or CH 2 , wherein V and U cannot be simultaneously O; L is a five or six membered heteroaryl group, selected from or to a pharmaceutically acceptable salt or acid addition salt, to a racemic mixture, or to its corresponding enantiomer and/or optical isomer and/or stereoisomer thereof. The compounds may be used for the treatment of Parkinson's disease, anxiety, emesis, obsessive compulsive disorder, autism, neuroprotection, cancer, depression and diabetes type 2.
priorityDate 2015-07-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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