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filingDate 2016-06-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eb2c4787dc1fc16679f4420fa0cb395a
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publicationDate 2018-04-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3302482-A1
titleOfInvention Tank-binding kinase-1 protacs and associated methods of use
abstract The present invention relates to bifunctional compounds, which find utility to degrade and (inhibit) TBK l. In particular, the present invention is directed to compounds, which contain on one end an E3 ubiquitin ligase binding moiety which binds to an E3 ubiquitin ligase and on the other end a moiety which binds TBKl such that TBKl is placed in proximity to the ubiquitin ligase to effect degradation (and inhibition) of TBKl. The present invention exhibits a broad range of pharmacological activities associated with compounds according to the present invention, consistent with the degradation/inhibition of TBKl.
priorityDate 2015-06-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4193
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7978
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126756
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395280
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP37237
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11683
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415878610
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID553788
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394128
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373125
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419586768
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1643
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8737
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419574085
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9PJN6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2187
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID15251
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QZU9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C0G6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506090
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397820
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID534935
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C0G7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409697
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP97712
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2XNF5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID441203
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO74810
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152743293
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID33032
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396823
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426106212
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID554230
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO74201
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419584733
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID19766
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419505924
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO74196
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10690
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426109678
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID85702142
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID53556
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397641
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06104
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393724
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421328696
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID317743
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393698
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ01651
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5833
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9876378
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399253
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID85702122
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100209445
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399254
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C236
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6P073
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID15211
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID58918
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID153274749
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393662
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419585571

Total number of triples: 1981.