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filingDate 2015-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_180713006a1ae3874df7835f10967afe
publicationDate 2016-12-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3109237-A1
titleOfInvention Novel 5-ht2 antagonists
abstract The present invention relates to 1-amidino-3-aryl-2-pyrazoline derivatives of the general formula In n The invention specifically relates to such derivatives which exhibit antagonizing activity towards serotonin 5-HT 2B receptors. The present invention also relates to use of said compounds as a medicament and for the treatment of fibrosis, cardiovascular diseases, pain, IBD, and other inflammatory diseases, as well as pharmaceutical compositions comprising one or more of said compounds and methods of treatment.
priorityDate 2015-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420237935
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393712
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12210218
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100136689
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Total number of triples: 730.