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filingDate 2015-02-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_02943e1e7b12a5470099611546249e49
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publicationDate 2016-12-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3103453-A1
titleOfInvention Medicinal composition comprising diamino heterocyclic carboxamide compound as active ingredient
abstract [Problem] To provide: a medicinal composition for treating an AXL-related cancer; in another embodiment, a medicinal composition for treating a cancer with high expression of AXL; and, in still another embodiment, a medicinal composition for treating a cancer that has acquired resistance through activation of AXL against anticancer agent therapy. [Solution] As the results of an examination on compounds having AXL inhibitory effect, the present inventors confirmed that specific diamino heterocyclic carboxamide compounds have AXL inhibitory effect and medicinal compositions comprising such a compound as an active ingredient have therapeutic effect on an AXL-related cancer, on a cancer with high expression of AXL in another embodiment, and on a cancer that has acquired resistance through activation of AXL against anticancer agent therapy in still another embodiment, thereby completing the present invention.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10744134-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3372231-A4
priorityDate 2014-02-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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