http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3095781-A1

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filingDate 2015-01-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_67bb1a0d4370d8412f182eaf2d5d8aef
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6b816211cb0a629cfbbcbd1e2d32d459
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1c1bf2d31eaaa6101495cb874b46c00e
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publicationDate 2016-11-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3095781-A1
titleOfInvention Indole compound
abstract [Problem] To provide a compound useful as a MT 1 and/or MT 2 receptor agonist. [Solution] The present inventors have studied on MT 1 and/or MT 2 receptor agonists, and have confirmed that indole compounds have the activity. As a result, the present invention is accomplished. That is, a compound represented by formula (I) or a salt thereof according to the present invention has a MT 1 and/or MT 2 receptor agonistic activity and has a low ability of migrating into the central nervous system. Therefore, the compound or a salt thereof can be used as a peripheral MT 1 and/or MT 2 receptor agonist, and therefore can be used as a therapeutic and/or prophylactic agent for urinary incontinence, particularly stress urinary incontinence and mixed urinary incontinence.
priorityDate 2014-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 506.