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filingDate 2014-09-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a6b1114c033450e0b9664281a9ea4e91
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_28eabf0bad81199082c4abe4e645ed3e
publicationDate 2016-07-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-3046591-A1
titleOfInvention S-enantiomer of tetracyclic indole derivative as pbr ligands
abstract The present invention concerns in vivo imaging and in particular in vivo imaging of translocator protein (TSPO, formerly known as the peripheral benzodiazepine receptor). An indole-based in vivo imaging agent is provided that overcomes problems relating to known TSPO-binding radiotracers. The present invention also provides a precursor compound useful in the synthesis of the in vivo imaging agent of the invent ion, as well as a method for synthesis of said precursor compound. Other aspects of the invention include a method for the synthesis of the in vivo imaging agent of the invention comprising use of the precursor compound of the invention, a kit for carrying out said method, and a cassette for carrying out an automated version of said method. In addition, the invention provides a radiopharmaceutical composition comprising the in vivo imaging agent of the invention, as well as methods for the use of said in vivo imaging agent.
priorityDate 2013-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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