http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2934529-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_0bddb695331af9b1a351ec38b1476e85
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-48
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filingDate 2013-12-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_49a96dcd8abddb1beeba74ae17c986cd
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eca01b541fe452d993c4a1128f1e3bcf
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2bdc17e763ac88567f0f4efef7aee9d6
publicationDate 2015-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2934529-A1
titleOfInvention Novel ergoline derivatives and uses thereof
abstract Provided herein are 8'-Hydroxy-2-CF3-dihydroergotamine (8 ' OH-2-CF3 -DHE) compounds, compositions, and dosage forms containing such compositions. Also provided herein are methods of treatment, prevention, or amelioration of a variety of medical disorders such as, for example, migraine using the compounds and compositions disclosed herein. In still other embodiments, provided herein are methods of agonizing receptors such as, for example, the 5-HT1D and/or the 5-HT1B receptor, without agonizing the 5-HT2B receptor using the compounds and compositions disclosed herein. In still other embodiments, provided herein are methods of antagonizing or inhibiting activity at receptors such as, for example, the adrenergic alpha2A and/or the alpha2B receptors using the compounds and compositions disclosed herein.
priorityDate 2012-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 749.