http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2881391-A1

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filingDate 2013-12-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2015-06-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2881391-A1
titleOfInvention Spiroindoline carbocycle derivatives and pharmaceutical compositions thereof
abstract Spiroindoline carbocycle derivatives, process for their preparation and pharmaceutical compositions thereof, their use for the treatment and/or prophylaxis of diseases, and their use for the manufacture of medicaments for the treatment and/or prophylaxis of diseases, especially sex-hormone-related diseases in both men and women, in particularly those selcted from the group of endometriosis, uterine fibroids, polycystic ovarian disease, hirsutism, precocious puberty, gonadal steroid-dependent neoplasia such as cancers of the prostate, breast and ovary, gonadotrope pituitary adenomas, sleep apnea, irritable bowel syndrome, premenstrual syndrome, benign prostatic hypertrophy, contraception and infertility (e.g., assisted reproductive therapy such as in vitro fertilization). The present application relates in particular to spiroindoline derivatives as gonadotropin-releasing hormone (GnRH) receptor antagonists.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311536446
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128054157
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129370350
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128354088
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118113136

Total number of triples: 618.