http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2751095-A2

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D243-12
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filingDate 2012-08-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bcebdb71c7855772690a785afecd2a2c
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7fb465fee5ccbe9a536edd85281ff3b3
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publicationDate 2014-07-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2751095-A2
titleOfInvention Novel benzodiazepinones as modulators of metabotropic glutamate receptor functions and neurological uses thereof
abstract The present invention relates to novel benzodiazepinone compounds of Formulae (I) wherein R 1 , R 2 , R 4 , R 6 , R 7 , R 8 , R 9 , and R 10 are as defined herein. The invention also relates to pharmaceutical compositions containing such compounds, methods of use of such compounds and compositions, and methods for preparing the compounds and compositions. The compounds are Group II metabotropic glutamate antagonists or allosteric modulators and are useful for the treatment of a variety of CNS disorders.
priorityDate 2011-08-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 892.