http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2729449-A1

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filingDate 2012-07-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_536e0d19e8bf468eed878db2b12f5305
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3883dfef7bceab720b6e18b4da94b8da
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_912e310fd7e1ff6ae775b0104d96ac21
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9e8e8082fca983c930a9b92dc3c3dc8e
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0bba564dc75c2a4bc446893b9c9d0d09
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b9d6e8940959b66f3c9891fe2fb54698
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_dc5a1ad1f52b90257b955b43cf30328a
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3b877f2895be5d86d0ea4d7a50929990
publicationDate 2014-05-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2729449-A1
titleOfInvention 5- or 6 - substituted 3 - hydroxy - 2 ( 1h) - pyridinones as d-amino acid oxidase (daao) inhibitors in therapy of diseases such as schizophrenia, cognitive disorder and pain
abstract The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof, wherein R 1 is hydrogen or fluorine, one of A and B is R2, the other is a group -X-Y-R3. R3 represents a carbocyclic or heterocyclic ring. Further variables are as defined in the specification. Also claimed are- processes for their preparation, pharmaceutical compositions containing them and their use in therapy of diseases such as schizophrenia, cognitive disorders and pain by modulating the D-amino acid oxidase enzyme (DAAO).
priorityDate 2011-07-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1408.