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filingDate 2011-07-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2013-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2596122-A2
titleOfInvention Modulators for sirt5 and assays for screening same
abstract Sirt5, a mitochondrial Sirtuin, has been identified herein as an efficient demalonylase and desuccinylase. Disclosed herein are assays to identify Sirt5 modulators based on this robust enzymatic activity. Sirt5-specific modulators can be used study the biological function of Sirt5 and to target Sirt5 activities in treating human diseases.
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