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publicationDate 2012-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2444120-A1
titleOfInvention Spirocyclic amiloride analogues as ENac blockers
abstract A compound of Formula In nin free or salt or solvate form, where R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R 9 , R 10 and R 11 have the meanings as indicated in the specification, is useful for treating diseases which respond to the blockade of the epithelial sodium channel. Pharmaceutical compositions that contain the compounds and processes for preparing the compounds are also described.
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Total number of triples: 2135.