http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2399921-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_28e3113097dd6d28720572e47f2f2407
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-04
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4545
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-444
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-437
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D513-04
filingDate 2009-11-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5e31d7ae22c8e7981bbf4406edb17c86
publicationDate 2011-12-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2399921-A1
titleOfInvention Heterocyclic compound and use thereof
abstract A compound represented by formula (I) or a salt thereof, which has a potent Raf inhibitory activity.n nIn formula (I), R 1 represents an optionally substituted C 1-6 alkyl, etc.; X represents -O- or -NR 2 - (wherein R 2 represents a hydrogen atom or a C 1-6 alkyl); Y represents a group represented by formula 2 (2i or 2ii)n n(wherein ring A represents an optionally substituted benzene ring; Z represents a group represented by (1) -NR 3 CO-W 1 -, (2) - NR 3 CO-W 1 -O-, (3) -NR 3 CO-W 1 -O-W 2 -, (4) -NR 3 CO-W 1 -S-, (5) -NR 3 CO-W 1 -NR 4 -, (6) -NR 3 COO-, (7) -NR 3 COO-W 1 -, (8) -NR 3 CO-CO-, or (9) - NR 3 CONR 4 - (wherein R 3 and R 9 each represents a hydrogen atom, etc., and W 1 and W 2 each represents an optionally substituted C 1-6 alkylene, etc.); and R 5 represents an optionally substituted five- or six-membered ring group.
priorityDate 2008-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 2455.