http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2380597-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_17832f1285ef628523e702754592582a |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K51-088 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K51-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K7-64 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K51-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K7-64 |
| filingDate | 2010-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4e338f12030861cd2f16908bf34a718e http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c02c7fb6b691ad29e8170cb6f37187c9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b4445e42cdca75cbfba81f0acc210cda http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c92d49cd275d387dd184baae98b05b9c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ab42fa5f611aba893cb58f0a1f3ffb5c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a4fcbcfb71bdf376c1080bcae36ab0da |
| publicationDate | 2011-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | EP-2380597-A1 |
| titleOfInvention | Cyclopeptide derivatives and uses thereof |
| abstract | The invention relates to compounds having a structure according to formula (I), cyclo[(R 1 )Xaa 1 -B-(R 2 )Xaa 2 -(R 3 )Xaa 3 -(R 4 )Xaa 4 ], or pharmaceutically acceptable salts thereof, wherein Xaa 1 and Xaa 3 are independently of each other, a natural or unnatural amino acid, preferably with Xaa 1 and Xaa 3 being, independently of each other, an amino acid comprising an aromatic moiety in its side chain, Xaa 2 is a natural or unnatural basic amino acid, Xaa 4 is glycine or a D-amino acid, R 1 , R 2 , R 3 and R 4 are independently of each other H or methyl, B is an amino acid group having a structure according to formula (II), -N(-Q)-CHR 5 -C(=O)-, wherein R 5 is selected from the group consisting of H, optionally substituted alkyl, optionally substituted aryl and optionally substituted heteroaryl, and a moiety L, and wherein Q is a group being sterically more demanding than a methyl group. The invention also relates to compositions, methods and uses related to said compounds. |
| priorityDate | 2010-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 550.