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filingDate 2003-04-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_29aee2f1bdff44d5b6f0937e27776b13
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publicationDate 2011-06-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2339347-A1
titleOfInvention Method of identifying transmembrane protein-interacting compounds
abstract A method for screening a candidate compound for its ability to interact with at least one transmembrane protein comprising: ntransfecting a cell with at least one nucleotide sequence encoding a protein comprising a transmembrane protein containing at least one nuclear localisation sequence (NLS) and a detectable moiety and permitting expression of the encoded protein in the cell; ncontacting the cell with a candidate compound; and ndetermining the distribution of the expressed protein in the cell by detecting the distribution of the detectable moiety in the cell; nwherein detection of an altered distribution of the detectable moiety in the cell relative to the distribution of the detectable moiety in a control cell not contacted with the candidate compound indicates that the compound interacts with the transmembrane protein, and nwherein the wild type transmembrane protein contains an NLS.
priorityDate 2002-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24827
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID37455
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8MI73
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100136153
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID843095
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2VHN8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9NS75
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID490404
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419485969
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4020
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226426779
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403993
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID268934
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID443006
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11839
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397491
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID497672
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400268
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID170926
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24318
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GL67
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP61279
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127443804
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49157
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ01631
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397554
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GL60
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3007
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID681
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49151
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09476
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GKR0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID404002
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5311080
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GKA2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81025
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393691
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24337
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100471532
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID821960
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1491913
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ866F4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09537
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226412710
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81071
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18610
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26617
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5PJB2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57282044
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09477
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP63296
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24329
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A1A7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP17647
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GMB3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GMB2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ867B1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24336
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24335
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1JI86
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO52629
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400187
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415749640
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100689321
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP63298
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554314
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A286ZRT7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP15208
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP63297
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16132283
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID436607
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A1A8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100722663
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81423
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID10800
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76L34
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5173
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3645
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4686
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0TKT1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395909
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO52847
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP50412
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1P4F9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76L33
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3643
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID252590
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ924T8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100136733
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID136083758

Total number of triples: 1054.