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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_0838837af9ee68143990bc0ce7b7838b
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-00
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K38-08
filingDate 2009-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d9f690125c2aea96241369eba11c8a59
publicationDate 2011-03-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2297179-A1
titleOfInvention Peptide analogues, particularly for the treatment of chronic pain
abstract The use is claimed of opioid peptides with a novel structure, which in addition to the pharmacophore contain structural elements that interact with neurotensisn receptors. Due to the synergistic interaction with the additional element, an augmented analgesic activity is obtained, capable of being used for an extended period due to decreased drug tolerance induction. These compounds may be of particular use in the treatment of chronic pain as effective analgesics during inflammation caused by rheumatoid, gout, neurodegeneration, post-operative or post-accidental lesions, or oncogenic lesions.
priorityDate 2008-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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