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filingDate 2005-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5a4b015cc54b9411f2e38c6408bb1dad
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publicationDate 2010-06-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2196469-A1
titleOfInvention Conjugates with anti-inflammatory activity
abstract The present invention relates to new compounds represented by Formula I: nwherein M represents a macrolide subunit of the substructure VIII: nL represents the chain of the substructure IX or XIII: n€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ -X 1 -(CH 2 ) m -Q-(CH 2 ) n -X 2 -€ƒ€ƒ€ƒ€ƒ€ƒIX n€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ -X 1 -(CH 2 ) m -V-(CH 2 ) p -Q-(CH 2 ) n -X 1 -€ƒ€ƒ€ƒ€ƒ€ƒXIII nZ represents the steroid or nonsteroidal subunit derived from steroid or nonsteroidal (NSAID) drugs with anti-inflammatory activity; The present invention relates also to pharmaceutically acceptable salts and solvates of such prepared compounds, to processe and intermediates for their preparation, as well as to the improved therapeutic action and the use in the treatment of inflammatory diseases and conditions in humans and animals.
priorityDate 2004-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5754
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57417230
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5753
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129783076
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Total number of triples: 1344.