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filingDate 2008-06-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2010-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5b364cc9d821f2739a7e1317b6b4956a
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eb6af49a06c853396e41d643a0cbe013
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publicationDate 2010-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2167046-B1
titleOfInvention Pharmaceutical solid preparation comprising benzazepines and production method thereof
abstract The subject invention provides a novel pharmaceutical solid preparation that has superior disintegration properties and excellent solubility, leading to sufficient absorbability of active ingredients through the gastrointestinal tract. The pharmaceutical solid preparation of the present invention comprises: (a) 7-chloro-5-hydroxy-1-[2-methyl-4-(2-methylbenzoylamino)benzoyl]-2,3,4,5-tetrahydro-1H-benzoazepine and/or salt thereof; (b) hydroxypropylcellulose containing a hydroxypropoxyl group in an amount of 50 wt.% or greater; and (c) at least one member selected from the group consisting of carmellose, sodium carboxy methyl starch, crospovidone, and low substituted hydroxypropylcellulose with an average particle diameter of 30 to 70µm, and a 90% cumulative particle diameter of 100 to 200µm.
priorityDate 2007-06-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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