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filingDate 2008-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2009-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2138507-A1
titleOfInvention Method for producing intermediates for the production of novel macrocycles that are inhibitors of the proteasomic degradation of p27, such as argyrin and derivatives thereof, and uses of said macrocycles
abstract The present invention relates to the use of particular macrocycles that are inhibitors of the proteasomic degradation of p27, in particular argyrin and derivatives thereof, for a treatment in a variety of conditions, such as the induction of immunotolerance, autoimmune diseases, bacterial infections, and proliferative diseases, such as cancers.
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