http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2044051-A1

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filingDate 2007-06-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e068782ce7d08c388b6291415df6cd5e
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publicationDate 2009-04-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2044051-A1
titleOfInvention Pyridine and pyrazine derivatives as mnk kinase inhibitors
abstract The present invention relates to compounds of the general formula (I) wherein X, Y, Z, A, Ar, R1, R2, R3, and R4 are as defined herein, which compounds are inhibitors of MNK2 and MNK1. The invention also relates to the use of the compounds in therapy, pharmaceutical compositions comprising the compounds, and the use of the compounds for the preparation of a medicament for the prophylaxis and treatment of disorders related to undesired activity of MNK1 and/or MNK2 kinases.
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priorityDate 2006-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129811210
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129355692
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403625
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24760312
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP29335
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Total number of triples: 1936.