http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2003120-A1

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filingDate 2008-06-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8b27687302d29d329d516f372c071f14
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publicationDate 2008-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2003120-A1
titleOfInvention Azapeptide derivatives as HIV protease inhibitors
abstract This invention relates to novel compounds of the Formula Ib:n nthat are azapeptides, and pharmaceutically acceptable salts thereof. More specifically, the invention relates to novel azapeptide compounds that are derivatives of the HIV protease inhibitor atazanavir sulfate. This invention also provides pyrogen-free compositions comprising one or more compounds of the invention and a carrier, and the use of the disclosed compounds and compositions in methods of treating diseases and conditions that are treated by administering HIV protease inhibitors. The invention also relates to the use of one or more of the disclosed compounds as reagents in analytical studies involving atazanavir.
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Total number of triples: 609.