http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1960356-A2

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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_85b084286a9881ef13644d09284d8c99
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publicationDate 2008-08-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1960356-A2
titleOfInvention Multivalent indole compounds and use thereof as phospholipase-a2 inhibitors
abstract Indole and indole-related compounds, compositions and methods are disclosed. The compounds of the invention are useful as phospholipase inhibitors. The compounds and compositions of the invention are useful for treatment of phospholipase- related conditions, such as insulin-related, weight-related and/or cholesterol-related conditions in an animal subject. The compounds of the invention consist of linked indole derivatives having at ' least two bicyclic rings of formula FIG. 6C in which R1R7 are defined as in claim 1 and in which the fused five membered ring contains a nitrogen atom and the fused six membered ring optionally contains one or two nitrogen atoms. The two or more bicyclic rings of Figure 6c are joined by a multifunctional bridge moiety substituted by two or more linking groups L which are joined to the bicyclic ring.
priorityDate 2005-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419571081
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JAX2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JAX3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09477
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100736962
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JAY0
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68549291
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410920896
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JAY1
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66021
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JAX9
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB02
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB03
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0JB00
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP80003
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09687
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Total number of triples: 2044.