http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1928826-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00
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filingDate 2006-09-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_485518ae0f2960478836fac35b4a84eb
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_92fbf5e481c421a14325fd1c0dd6ae86
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_aa297a20c9b53eb5d0bf7e7e4fe16a39
publicationDate 2008-06-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1928826-A1
titleOfInvention Sulphonylpyrrole hydrochloride salts as histone deacetylases inhibitors
abstract Compounds of formula I, in which R1, R2, R3, R4, R5, R6 and R7 have the meanings indicated in the description, as well as salts thereof are novel effective HDAC inhibitors. In more detail, this invention refers to salts of a compound selected from (E)-(E)-N-hydroxy-3-(1-[4-(([2-(1H-indol-2yl)-ethyl]-methyl-amino)-methyl)-benzene sulfonyl]-1H-pyrrol-3-yl)-acrylamide, (E)-3-[1-(4-dimetylaminomethyl-benzenesulfonyl)-1H-pyrrol-3-yl]-N-hydroxy-acrylamide, and (E)-N-hydroxy-3-[1-(5-pyridin-2-yl-thiophene-2-sulfonyl)-1H-pyrrol-3-yl]-acrylamide with hydrochloric acid, their hydrates and to crystalline forms of these salts and hydrates.
priorityDate 2005-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 2005.