http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1925295-A1

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filingDate 2006-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2008-05-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1925295-A1
titleOfInvention Stable powder formulation containing a new antichinolinergic agent
abstract The present invention relates to a spray-dried powder formulation comprising particles which contain the following components i) to iii): i) anticholinergics, especially at least one compound of formula 1 wherein X - a negatively charged anion means ii) at least one embedding material selected from the group consisting of mono- or disaccharides, oligosaccharides, polymers, sugar alcohols and cholesterol, iii)) an organic, physiologically acceptable, sterically demanding acid selected from the group consisting of ascorbic acid, a mono-, di- or trihydric carboxylic acid with the exception of aminocarboxylic acids, preferably fumaric acid, oxalic acid or succinic acid, and a fruit or edible acid, preferably citric acid , Tartaric acid, malic acid, lactic acid, acetic acid, α-hydroxycaproic acid or gluconic acid, a process for their preparation, and the use of an organic, physiologically harmless, sterically demanding acid from the group consisting of ascorbic acid, a mono-, di- or trihydric carboxylic acid, with the exception of aminocarboxylic acids, preferably fumaric acid, oxalic acid or succinic acid, and a fruit or edible acid, preferably citric acid, tartaric acid, malic acid, lactic acid, acetic acid, α-hydroxycaprylic acid or gluconic acid, for stabilizing a spray-dried powder formulation comprising the above compound of formula 1 according to i) and a suitable embedding material ii).
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2023187393-A1
priorityDate 2006-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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