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filingDate 2006-03-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2009-05-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e5a56ce115a1590041df724378ccd4d0
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6ec40a8c41cacc74852a57df82563c69
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publicationDate 2009-05-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1866286-B1
titleOfInvention Pyridine derivatives useful as inhibitors of pkc-theta
abstract Disclosed are novel compounds of formula (I) wherein R1, R2 and R3 are as defined herein, which are useful as inhibitors of PKC-theta and are thus useful for treating a variety of diseases and disorders that are mediated or sustained through the activity of PKC-theta, including immunological disorders and type II diabetes. This invention also relates to pharmaceutical compositions comprising these compounds, methods of using these compounds in the treatment of various diseases and disorders, processes for preparing these compounds and intermediates useful in these processes.
priorityDate 2005-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95KV1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2MVY4
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ32KY4
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95KV0
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453706522
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2756045
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12275765
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227849312
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58712686
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID245803200
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163498731
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129765641
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2724994
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60328
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID977
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58712687
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP15208
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID609429
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58712689
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119411
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP05412
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID48311
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Total number of triples: 411.