http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1858509-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-04
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-415
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filingDate 2006-03-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fd2ebf4ce2051cf2d509d8320a9a12ee
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8a38079d72bb4463404d98d657a2f741
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_071ca58519567b584e02f84cb33ae7e6
publicationDate 2007-11-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1858509-A1
titleOfInvention Novel cathepsin c inhibitors and their use
abstract The invention is directed to novel cathepsin C inhibitors and their use in the treatment of diseases mediated by the cathepsin C enzyme. Specifically, the invention is directed to compounds according to Formula (I): wherein X and n are defined below, and to pharmaceutically-acceptable salts thereof. The compounds of the invention are cathepsin C inhibitors and can be used in the treatment of diseases mediated by the cathepsin C enzyme, such as COPD. Accordingly, the invention is further directed to pharmaceutical compositions comprising a compound of the invention. The invention is still further directed to methods of inhibiting cathepsin C and treatment of conditions associated therewith using a compound of the invention or a pharmaceutical composition comprising a compound of the invention.
priorityDate 2005-03-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 615.