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filingDate 2005-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_34ec7d5346d3f5724431da749a9fee2a
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publicationDate 2007-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-1752544-A1
titleOfInvention Probe for detecting nuclear receptor agonist or antagonist and method of screening agonist or antagonist to nuclear receptor with the use of the same
abstract A probe for detecting an agonist or an antagonist to a nuclear receptor, in which, at least, a ligand-recognition site containing a ligand-binding domain of the nuclear receptor is connected with a binding-responsive site containing a peptide chain that specifically binds to a coactivator-binding site in the ligand-binding domain by a flexible linker to construct a fusion structure [ligand-recognition site/linker/binding-responsive site], and two reporters are connected with the respective ends of the fusion structure.
priorityDate 2004-02-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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