http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1742957-B1
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_81075572b8d1526ce20dbf5dd7dbded8 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07H17-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07H17-08 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07H17-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07H17-00 |
filingDate | 2005-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate | 2007-09-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_037da872be2a8dc7a18cf5eee8b2e3f5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6e1e419800a974ef6df02b60387e65e7 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0f36e01e82a3bf2c168513a29dbd91f3 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_01b493ab025ca064453961d63531df1c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_220b10dc5cdcedb254b87f5d12f7ac05 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6d339a4957e441ca5c708eafd2cda6a7 |
publicationDate | 2007-09-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | EP-1742957-B1 |
titleOfInvention | Process for the preparation of telithromycin |
abstract | The present invention relates to the process for the preparation of compounds of formula (I) or its pharmaceutically acceptable salts Formula I The novel compounds (i) 10,11-Anhydro-2',4''-di-O-benzoyl-12-O-imidazolylcarbonyl-6-O-methylerythromycin A of formula (Xa) Formula (Xa) (ii) 2',4''-di-O-benzoyl-11-amino-11-N-[4-[4-(3-pyridyl)imidazol-1-yl]butyl]-11-deoxy-6-O-methylerythromycin A 11,12-cyclic carbamate of formula (XIa) Formula (XIa) (iii) 2'-O-benzoyl-11-amino-11-N-[4-[4-(3-pyridyl)imidazol-1-yl]butyl]-11-deoxy-5-O-desosaminyl-6-O-methylerythronolide A 11,12-cyclic carbamate of formula (XIIa) Formula (XIIa) (iv) 2'-benzoyl-11-amino-11-N-[4-[4-(3-pyridyl)imidazol-1-yl]butyl]-11-deoxy-5-O-desosaminyl-6-O-methylerythronolide A 11,12-cyclic carbamate of formula (XIIa) Formula (XIIa) and their use as intermediates in formation of compound of Formula I. Also the process of preparation of compound of formula (XIIIa). Formula (XIIIa) |
priorityDate | 2004-04-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 135.